Term Name: PF-3758309
Synonyms: N-[(1S)-2-(dimethylamino)-1-phenylethyl]-6,6-dimethyl-3-[(2-methylthieno[3,2-d]pyrimidin-4-yl)amino]-4,6-dihydropyrrolo[3,4-c]pyrazole-5(1H)-carboxamide, PF 309, PF 3758309, PF-03758309, PF-309, PF309, PF3758309
Definition: A member of the class of thienopyrimidines that is thieno[3,2-d]pyrimidine substituted by methyl and (5-{[(1S)-2-(dimethylamino)-1-phenylethyl]carbamoyl}-6,6-dimethyl-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl)amino groups at positions 2 and 4, respectively. It is a potent inhibitor of PAK4 and inhibits the growth of multiple human tumor xenografts.
Ontology: ChEBI [CHEBI:93751]  ( EBI )

Relationships
is a type of: benzenes pyrrolopyrazole secondary amino compound tertiary amino compound thienopyrimidine ureas
has_role: antineoplastic agent apoptosis inducer EC 2.7.11.1 (non-specific serine/threonine protein kinase) inhibitor